Product Details: Alarelin Acetate

Alarelin acetate is a synthetic peptide analog of gonadotropin-releasing hormone (GnRH) used in laboratory research to study endocrine regulation. It belongs to the class of GnRH agonists and has been investigated in experimental systems involving reproductive and hormonal signaling. [1][2]

Mechanism of Action

Alarelin acetate functions as a GnRH receptor agonist by interacting with receptors on anterior pituitary gonadotroph cells, leading to the release of luteinizing hormone (LH) and follicle-stimulating hormone (FSH) in experimental systems. [2][4]

GnRH receptor activation is known to involve intracellular signaling pathways such as phospholipase C activation and calcium mobilization. These pathways are widely studied in GnRH-related research to understand hormone secretion dynamics. [3]

Prolonged or repeated stimulation of GnRH receptors is associated with receptor desensitization and reduced gonadotropin release. This biphasic response is a characteristic feature of GnRH agonist activity and is used in experimental models to study endocrine regulation and feedback mechanisms. [3]

Properties of Alarelin Acetate:

• Molecular Formula: C60H86N16O16
• Molecular Weight: 1287.4 g/mol
• CAS Number: 79561-22-1
• PubChem CID: 12821051
• Synonyms: 288L2XKV2J, LHRHa, RefChem:1076311, Leutenizing Hormone-Releasing Hormone analogue

Research Applications/Benefits of Alarelin Acetate

• GnRH Receptor Activation Studies

Alarelin is used in laboratory models to study GnRH receptor binding and signaling pathways. [2]

• Gonadotropin Secretion Research

It supports studies investigating LH and FSH release and pituitary signaling dynamics. [2][4]

• Endocrine Feedback and Desensitization Models

Alarelin is applied in experimental systems examining receptor regulation and hormonal feedback responses associated with GnRH signaling. [3]

• Reproductive Endocrinology Studies

It is used in research involving HPG axis regulation and reproductive hormone signaling. [2][4]

Why Choose BehemothLabz for Alarelin Acetate?

Choose BehemothLabz, choose quality! We are among the few online sellers that believe in the integrity and purity of products. Our Alarelin Acetate is designed to meet the industrial criteria and the needs of researchers. Before launching our products, we test them through an independent laboratory to check their purity and ingredients. This procedure maximizes the accuracy and findings of your research experiments.  

Additionally, we deliver nationwide and internationally. We use a secure payment system that safeguards your personal information and prevents unauthorized third-party access.

So, purchase Alarelin acetate now and experience quality and purity for your research.

Disclaimer: This information is for educational purposes. We do not allow the human consumption of our products. All our products are sold for laboratory and research experiments. 

References

1. Yuan, F., Zhang, P., Liu, M., Li, Y., Xu, B., & Li, X. (2025). Pharmacogenomic analysis of alarelin acetate-induced hepatotoxicity: a case report and literature review. Frontiers in Medicine, 12, 1634101. 
2. Yang, H., Huang, G., Lv, M., Lin, Y., Wang, R., Zeng, L., Ma, H., & Hu, T. (2018). Immune Effects of Alarelin on Ovarian Development and GnRH Receptor mRNA Expression Levels of the pituitary in tilapia (Oreochromis niloticus). Turk. J. Fish. & Aquat. Sci., 19(4), 289–296. 
3. Naor, Z., Harris, D., & Shacham, S. (1998). Mechanism of GNRH receptor signaling: combinatorial Cross-Talk of Ca²⁺ and protein kinase C. Frontiers in Neuroendocrinology, 19(1), 1–19. 
4. Wei, S., Chen, S., Gong, Z., Ouyang, X., An, L., Xie, K., Dong, J., & Wei, M. (2013). Alarelin active immunization influences expression levels of GnRHR, FSHR and LHR proteins in the ovary and enhances follicular development in ewes. Animal Science Journal, 84(6), 466–475.