Cardarine GW 501516 Liquid

Cardarine GW-501516, often associated with SARMs, is a PPARδ agonist. Peroxisome Proliferator-Activated Receptor Delta (PPARδ) agonist. It has been shown in preclinical models to upregulate mitochondrial biogenesis and enhance fatty acid oxidation.

PPARδ has been investigated for its potential involvement in lipid metabolism, skeletal muscle physiology, and cardiovascular function. Additionally, studies in experimental models have shown its role in glycemic regulation and muscle cell signaling pathways.

Working Mechanism of Cardarine GW-501516 Liquid

Cardarine works in a similar pattern to GW0742. It activates PPARδ receptors in experimental models, which in turn potentially perform a key role. Activation of these receptors has been studied for its role in regulating metabolic pathways, particularly those associated with fatty acid oxidation and energy homeostasis. These mechanisms are being investigated for their involvement in metabolic research contexts.

Properties of Cardarine GW-501516

• Chemical Formula: C21H18F3NO3S2
• Synonym: GW-501,516
• IUPAC-Name: 2-[2-methyl-4-[[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]methylsulfanyl]phenoxy]acetic acid
• Molar Mass: 453.5 g/mol
• CAS Number: 317318-70-0
• PubChem CID: 9803963
• Shelf Life: 36 months

Research Findings on Cardarine 

Studies show how Cardarine, as a PPARδ agonist, influences lipid metabolism at the cellular level. In experimental models such as skeletal muscle cells, activation of PPARδ by GW-501516 has been shown to regulate the expression of genes involved in fatty acid oxidation and lipid utilization. These studies report increased activity of pathways linked to β-oxidation and energy metabolism. This suggests that the compound plays a role in shifting cellular energy use toward fatty acids rather than glucose. These findings highlight its relevance in metabolic pathway research, particularly in understanding lipid homeostasis and energy regulation.

Another research has examined the effects of GW-501516 on inflammatory and metabolic signaling pathways. In controlled cellular studies, activation of PPARδ by this compound has been observed to interfere with IL-6–mediated signaling, including suppression of STAT3 activation and related pathways associated with insulin resistance. These findings suggest that GW-501516 may influence molecular mechanisms linked to inflammation and cellular metabolic balance. However, such observations are limited to experimental models, and further investigation is required to fully understand these interactions.

Note: Cardarine is not approved by the FDA for any medical use. It remains an investigational compound and is made available for laboratory and research purposes only. It is not intended for human consumption.

Why Choose BehemothLabz to Buy Cardarine GW501516 Online?

We, Behemoth Labz, stand behind our Cardarine products and ensure that third-party-tested products reach our valued customers. Similarly, we offer competitive prices at discounted delivery charges with no compromise on the quality of the GW501516 products. 

Additionally, we also back our GW501516 products by providing excellent customer satisfaction. On top of that, we are among a few places that offers Cardarine for sale in capsules, liquid, and parenteral solution forms. 

Note: For a well-rounded research approach, explore our range of SARM Support products, designed to complement various research compounds. Additionally, check out Arimistane Liquid for potential estrogen regulation and Clomiphene for post-research applications. Enhance your research experience with BehemothLabz’s comprehensive selection of high-quality compounds.

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Reference Links

PubChem. (2026). GW 501516. Nih.gov; PubChem. https://pubchem.ncbi.nlm.nih.gov/compound/gw-501516

Dressel, U., Allen, T. L., Pippal, J. B., Rohde, P. R., Lau, P., & Muscat, G. E. O. (2003). The peroxisome proliferator-activated receptor beta/delta agonist, GW501516, regulates the expression of genes involved in lipid catabolism and energy uncoupling in skeletal muscle cells. Molecular Endocrinology (Baltimore, Md.), 17(12), 2477–2493. https://doi.org/10.1210/me.2003-0151

Serrano-Marco, L., Barroso, E., El Kochairi, I., Palomer, X., Michalik, L., Wahli, W., & Vázquez-Carrera, M. (2012). The peroxisome proliferator-activated receptor (PPAR) β/δ agonist GW501516 inhibits IL-6-induced signal transducer and activator of transcription 3 (STAT3) activation and insulin resistance in human liver cells. Diabetologia, 55(3), 743–751. https://doi.org/10.1007/s00125-011-2401-4