Cardarine (GW-501516) is an investigational small-molecule compound. It is classified as a PPARδ (Peroxisome Proliferator-Activated Receptor delta) agonist. 

In preclinical evaluations, Cardarine GW has been observed to act as a PPARδ (Peroxisome Proliferator-Activated Receptor Delta) agonist.  

Researchers believe that activation of PPARδ has been associated with potential changes in β-oxidation of fatty acids. It may also influence intracellular activity and homeostatic metabolic modulation in laboratory research models. 

However, these observations remain strictly limited to scientific research. Cardarine is not approved for human consumption.

BehemothLabz supplies Cardarine capsules exclusively for laboratory and investigational research.

Properties of Cardarine GW-501516

• Chemical Formula: C21H18F3NO3S2
• Synonym: GW-501,516, GW1516
• IUPAC-Name: 2-[2-methyl-4-[[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]methylsulfanyl]phenoxy]acetic acid
• Molar Mass: 453.5 g/mol
• CAS Number: 317318-70-0
• PubChem CID: 9803963
• Shelf Life: 36 months

How Does Cardarine 501516 Capsule Work?

Researchers have observed that Cardarine GW formulations may work similarly to GW0742 chemicals. They have the potential for ligand-binding interaction with PPARδ nuclear receptors in experimental models. 

After binding, GW formulations then potentially activate PPARδ to perform its key role in the research investigations.

The potential role of PPARδ may include alteration of adipogenic gene expression and upregulation of lipid catabolic processes.

Possible Research Applications of Cardarine 501516

Cardarine 501516 is an investigational compound that may have possible applications in the research field. A few of its potential applications that researchers have observed include:

• PPARδ activation studies are used to investigate receptor binding, activation, and downstream transcriptional regulation mechanisms.
• Substrate utilization pathway analysis is applied to examine shifts in lipid-associated versus glucose-associated biochemical signaling pathways.
• Oxidative pathway signaling research is utilized to study the regulation of pathways linked to mitochondrial-associated energy processes and endurance-related signaling dynamics.

Why Choose BehemothLabz to Buy Cardarine GW-501516?

Start your research today! Buy Cardarine now. If you are looking for a reasonable and high-quality Cardarine for sale, your search ends here. BehemothLabz offers Cardarine GW 501516 for sale to meet your research needs and industrial standards. 

You can verify lab results as each product batch gets a unique batch number. It is linked to a Certificate of Analysis (COA). The COAs are supposed to be accessible via product pages.

Behemoth Labz Disclaimer

All Behemoth Labz products are strictly for LABORATORY AND RESEARCH PURPOSES ONLY. They are not to be used for any human or veterinary purposes.

Please make sure you go through the Terms and Conditions and familiarize yourself with them, as they are important. Kindly research the scientific uses of this product before making any purchases. Make note that the packaging and labels of the product may differ from those shown on the website.

Buying the product means you agree to our Terms and Conditions. You can contact our customer service team at support@behemothlabz.com for queries.

Reference links

Turza, A., Bosca, M., Marieta Muresan-Pop, Mare, L., Gheorghe Borodi, & Popescu, V. (2025). Novel Solid Forms of Cardarine/GW501516 and Their Characterization by X-Ray Diffraction, Thermal, Computational, FTIR, and UV Analysis. Pharmaceutics, 17(2), 152–152. https://doi.org/10.3390/pharmaceutics17020152

Turza, A., Pascuta, P., Muresan-Pop, M., Mare, L., Borodi, G., & Popescu, V. (2024). Five Novel Polymorphs of Cardarine/GW501516 and Their Characterization by X-ray Diffraction, Computational Methods, Thermal Analysis, and a Pharmaceutical Perspective. Pharmaceutics, 16(5), 623. https://doi.org/10.3390/pharmaceutics16050623

Chen, W., Gao, R., Xie, X., Zheng, Z., Li, H., Li, S., Dong, F., & Wang, L. (2015). A metabolomic study of the PPARδ agonist GW501516 for enhancing running endurance in Kunming mice. Scientific Reports, 5(1). https://doi.org/10.1038/srep09884